1Department of Pharmaceutical Chemistry, K. M. College of Pharmacy, Uthangudi, Madurai -625107, Tamilnadu, India
2Department of Pharmacology, K. M. College of Pharmacy, Uthangudi, Madurai -625107, Tamilnadu, India
3Department of Pharmacognosy, K. M. College of Pharmacy, Uthangudi, Madurai -625107, Tamilnadu, India
4Department of Biochemistry, K. M. College of Pharmacy, Uthangudi, Madurai -625107, Tamilnadu, India
5Department of Biotechnology, St. Michael College of Engineering, Sivagangi, Tamilnadu, India
*Corresponding Author E-mail: meeraharsa@yahoo.com
Online published on 3 April, 2013.
Para substituted N-aryl anthranilic acid derivatives were synthesized via Ullmann condensation of o-Chlorobenzoic acid with various p-substituted aniline in the presence of cupric oxide (catalyst) and anhydrous potassium carbonate (for removal of hydrogen halide formed during reaction). The synthesized compounds (Ia-Ih) were evaluated the following biological activities Anti-inflammatory, Analgesic activity, Anti-bacterial activity. Organism used: Staphylococcus aureus (MTCC 96) Klebsiella aerogenes (MTCC), E. Coli (MTCC 722) Standard Used: Oflaxacin (10μg/disc)
N-aryl anthranilic acid derivative, Anti inflammatory, Analgesic, Anti bacterial